| Anticoagulants |
Vitamin K antagonists (inhibit II, VII, IX, X) |
coumarins: Acenocoumarol • Coumatetralyl • Dicoumarol (Dicumarol) • Ethyl biscoumacetate • Phenprocoumon • Warfarin
1,3-indandiones: Clorindione • Diphenadione • Phenindione
other: Tioclomarol |
Factor Xa inhibitors (with some II inhibition) |
Heparin group/ glycosaminoglycans/ (bind antithrombin) |
low molecular weight heparin (Bemiparin, Certoparin, Dalteparin, Enoxaparin, Nadroparin, Parnaparin, Reviparin, Tinzaparin)
oligosaccharides (Fondaparinux, Idraparinux)
heparinoid (Danaparoid, Sulodexide, Dermatan sulfate) |
| Direct factor Xa inhibitors |
xabans (Apixaban, Otamixaban, Rivaroxaban) |
|
| Direct thrombin (II) inhibitors |
bivalent: Hirudin (Bivalirudin, Lepirudin, Desirudin)
univalent: Argatroban • Dabigatran • Melagatran • Ximelagatran |
| Other |
Defibrotide • Ramatroban • Antithrombin III • Protein C (Drotrecogin alfa) |
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