Pethidine Intermediate A

Pethidine Intermediate A
	File:Pethidineintermediate.svg
Clinical data
Synonyms	Pethidine Intermediate A
Routes of; administration	N/A
Legal status
Legal status	US: Schedule I ;
Identifiers
	IUPAC name 1-methyl-4-phenylpiperidine-4-carbonitrile;
CAS Number	3627-62-1;
PubChem CID	62513;
E number	{{#property:P628}}
ECHA InfoCard	{{#property:P2566}}Lua error in Module:EditAtWikidata at line 36: attempt to index field 'wikibase' (a nil value).
Chemical and physical data
Formula	C13H16N2
Molar mass	200.28 g/mol

Pethidine Intermediate A is a 4-phenyl piperidine derivative that is a precursor to the opioid analgesic drug pethidine (meperidine). It is not known to have any analgesic activity in its own right, however other derivatives of pethidine with a 4-cyano group in place of the carboxylate ethyl ester have been found to be active,^[1] so Pethidine Intermediate A might also show opioid effects.

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References

↑ Lomenzo SA, Rhoden JB, Izenwasser S, Wade D, Kopajtic T, Katz JL, Trudell ML. Synthesis and Biological Evaluation of Meperidine Analogues at Monoamine Transporters. Journal of Medicinal Chemistry. 2005; 48:1336-1343.

Template:Opioids

[1] Lomenzo SA, Rhoden JB, Izenwasser S, Wade D, Kopajtic T, Katz JL, Trudell ML. Synthesis and Biological Evaluation of Meperidine Analogues at Monoamine Transporters. Journal of Medicinal Chemistry. 2005; 48:1336-1343.

[1]

Pethidine Intermediate A

References

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