Template:Affinities of selected androgen receptor ligands
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| Compound | AR RBA (%) | |
|---|---|---|
| Metribolone | 100 | |
| Dihydrotestosterone | 85 | |
| Cyproterone acetate | 7.8 | |
| Bicalutamide | 1.4 | |
| Nilutamide | 0.9 | |
| Hydroxyflutamide | 0.57 | |
| Flutamide | <0.0057 | |
| Note: Human prostate tissue used for the assays. Source: [1] | ||
References
- ↑ Ayub M, Levell MJ (August 1989). "The effect of ketoconazole related imidazole drugs and antiandrogens on [3H] R 1881 binding to the prostatic androgen receptor and [3H]5 alpha-dihydrotestosterone and [3H]cortisol binding to plasma proteins". J. Steroid Biochem. 33 (2): 251–5. doi:10.1016/0022-4731(89)90301-4. PMID 2788775.